Tilidine
Synthetic opioid painkiller / From Wikipedia, the free encyclopedia
Dear Wikiwand AI, let's keep it short by simply answering these key questions:
Can you list the top facts and stats about Tilidine?
Summarize this article for a 10 year old
SHOW ALL QUESTIONS
Tilidine, sold under the brand name Valoron among others, is a synthetic opioid analgesic, used mainly in Belgium, Bulgaria, Germany, Luxembourg, South Africa, and Switzerland for the treatment of moderate to severe pain, both acute and chronic.[4][5] Its onset of pain relief after oral administration is about 10–15 minutes and peak relief from pain occurs about 25–50 minutes after administration.[3]
Quick Facts Clinical data, Trade names ...
Clinical data | |
---|---|
Trade names | Valoron, others |
Other names | Tilidate (BAN UK) |
AHFS/Drugs.com | International Drug Names |
Routes of administration | Oral, rectal, IM, IV |
ATC code | |
Legal status | |
Legal status |
|
Pharmacokinetic data | |
Bioavailability | 6% (parent compound), 99% (active metabolite)[2] |
Metabolism | Metabolized by the liver, mostly via the enzymes CYP3A4 and CYP2C19[3] |
Elimination half-life | 3–5 hours[3] |
Excretion | Urine (90%)[3] |
Identifiers | |
| |
CAS Number | |
UNII | |
KEGG |
|
ChEBI | |
ChEMBL | |
ECHA InfoCard | 100.039.779 |
Chemical and physical data | |
Formula | C17H23NO2 |
Molar mass | 273.376 g·mol−1 |
3D model (JSmol) | |
| |
NY (what is this?) (verify) |
Close