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2C-B-morpholine

Pharmaceutical compound From Wikipedia, the free encyclopedia

2C-B-morpholine
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2C-B-morpholine, also known as 2C-B-norphenmetrazine or as 2-(4-bromo-2,5-dimethoxyphenyl)morpholine, is a serotonin receptor modulator of the phenylmorpholine (phenmetrazine) and cyclized phenethylamine groups.[1] It is a ligand of the serotonin 5-HT2A receptor, with an affinity of 20.6 nM and an EmaxTooltip maximal efficacy of 4%.[1] The drug showed 103-fold lower affinity for this receptor than R(–)-DOB and had minimal agonist activity (with R(–)-DOB having an Emax of 51% in the assay), so for practical purposes would act as an antagonist at the 5-HT2A receptor under most circumstances, despite being technically classified as a partial agonist.[1] 2C-B-morpholine was first described in the scientific literature by Richard Glennon and colleagues by 2004.[1]

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