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Bexirestrant
Chemical compound From Wikipedia, the free encyclopedia
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Bexirestrant is a selective estrogen receptor degrader (SERD) which is being evaluated for the treatment of breast cancer. This orally bioavailable compound has demonstrated potent activity against both wild-type and mutant forms of the estrogen receptor (ER), addressing a critical need in overcoming resistance to current endocrine therapies.[1]
It is structurally characterized by an E-alkene linked to an azetidine core.
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