Iferanserin

Iferanserin (INN; VEN-309) is a drug which acts as a selective 5-HT_2A receptor antagonist.^[1] It is under development as an intra-rectal formulation for the treatment of hemorrhoid disease, and as of February 2012, is in phase IIb clinical trials.^[1]

Iferanserin

Clinical data
ATC code	none
Identifiers
IUPAC name (E)-N-[2-[2-[(2S)-1-methylpiperidin-2-yl]ethyl]phenyl]-3-phenylprop-2-enamide
CAS Number	58754-46-4 Y
PubChem CID	6445539
ChemSpider	4949235
UNII	NWR3BEB8PA
ChEMBL	ChEMBL2107754
CompTox Dashboard (EPA)	DTXSID101030346
Chemical and physical data
Formula	C23H28N2O
Molar mass	348.490 g·mol−1
3D model (JSmol)	Interactive image
SMILES O=C(\C=C\c1ccccc1)Nc2ccccc2CC[C@H]3N(C)CCCC3
InChI InChI=1S/C23H28N2O/c1-25-18-8-7-12-21(25)16-15-20-11-5-6-13-22(20)24-23(26)17-14-19-9-3-2-4-10-19/h2-6,9-11,13-14,17,21H,7-8,12,15-16,18H2,1H3,(H,24,26)/b17-14+/t21-/m0/s1 Key:UXIPFQUBOVWAQW-UEBLJOKOSA-N